Progesterone receptor-Selectief Inhibitors | Agonists | Antagonists | Chemicals | Modulators

Estrogen receptor
Progesterone receptor

Cat.nr.	Productnaam	Informatie	Selectief / Pan	IC50 / Ki
S2606	Mifepristone	Mifepristone is a remarkably active antagonist of progesterone receptor and glucocorticoid receptor with IC50 of 0.2 nM and 2.6 nM, respectively.	Selective	Progesterone receptor, IC50: 0.2 nM
S2611	Ethisterone	Ethisterone is a progestogen hormone being considered to treat prostate cancer.	Selective
S1705	Progesterone	Progesterone is a C-21 steroid hormone.	Selective
S1304	Megestrol Acetate	Megestrol Acetate is a synthetic progesteronal agent with an IC50 of 260 μM for the inhibition of HepG2.	Selective
S3081	Ulipristal	Ulipristal is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure.	Selective
S3160	Ethynodiol diacetate	Ethynodiol diacetate is one of the first synthetic progestogens used in contraceptive pills.	Selective
S2567	Medroxyprogesterone acetate	Medroxyprogesterone acetate is a progestin, a synthetic variant of the human hormone progesterone and a potent progesterone receptor agonist.	Selective
s1251	Dienogest	Dienogest is an orally active synthetic progesterone, used for contraception and the treatment of endometriosis.	Selective
S1914	Pregnenolone	Pregnenolone is an endogenous steroid hormone for inhibition of M1 receptor- and M3 receptor-mediated currents with IC50 of 11.4 μM and 6.0 μM, respectively.	Selective
S4097	Dydrogesterone	Dydrogesterone is an orally active progestogen which acts directly on the uterus, producing a complete secretory endometrium in an estrogen-primed uterus.	Selective
S1377	Drospirenone	Drospirenone is a synthetic progestin that is an analog to spironolactone.	Selective
S3167	Altrenogest	Altrenogest is a progestogen structurally related to veterinary steroid trenbolone.	Selective
S1376	Gestodene	Gestodene is a progestogen hormonal contraceptive.	Selective
S1727	Levonorgestrel	Levonorgestrel is a synthetic progestogen used as an active ingredient in some hormonal contraceptives.	Selective